化合物GR 125743 T8737

Product Introduction
Bioactivity


英文名: GR 125743

描述: GR 125743 是选择性的5-HT1B/1D 受体拮抗剂，与野生型的人 h5-HT1B 和 5-HT1D 结合的pKi 分别为 8.85 和 8.31，可用于帕金森病和心血管疾病的研究。

体外活性: GR-125743, a new radiolabelled derivative of a compound that exhibits selective antagonistic properties with respect to the serotonin human (h5-HT1D) and human (h5-HT1B) receptors.?The compound has been characterized for its ability to label the cloned h5-HT1D and h5-HT1B receptors.

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 4.17 mg/mL (10 mM)


关键字: GR 125743 | h5-HT1B | cognitive disorder | h5-HT1D | cardiovascular | inhibit | Parkinson's disease | 5-HT Receptor | 5-hydroxytryptamine Receptor | receptor | Inhibitor | GR-125743 | Serotonin Receptor | GR125743

相关产品: Dexchlorpheniramine Maleate | Dasotraline hydrochloride | Jatrorrhizine | Mirtazapine D3 | BRL 54443 | Org 13011 | SAX-187 | Dolasetron Mesylate hydrate | (S)-Mirtazapine | AM9405

相关库: Anti-Neurodegenerative Disease Compound Library | Anti-Parkinson's Disease Compound Library | Angiogenesis related Compound Library | Anti-Cancer Compound Library | Membrane Protein-targeted Compound Library | Neuronal Signaling Compound Library | Inhibitor Library | GPCR Compound Library | Serotonin Receptor-Targeted Compound Library | NO PAINS Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途