化合物PFM01 T8880
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 1558598-41-6 | ¥1,270.00 | 询底价 |
50 mg | 1558598-41-6 | ¥2,320.00 | 询底价 |
5 mg | 1558598-41-6 | ¥398.00 | 询底价 |
200 mg | 1558598-41-6 | ¥4,730.00 | 询底价 |
100 mg | 1558598-41-6 | ¥3,730.00 | 询底价 |
1 mg | 1558598-41-6 | ¥186.00 | 询底价 |
1 mL | 1558598-41-6 | ¥448.00 | 询底价 |
10 mg | 1558598-41-6 | ¥663.00 | 询底价 |
Product Introduction
Bioactivity
英文名: PFM01
描述: PFM01 是 MRE11核酸内切酶抑制剂,是 N-烷基化的 Mirin 衍生物。它可以通过非同源末端连接 (NHEJ) 和同源重组 (HR) 调节双链断裂修复 (DSBR)。
体外活性: PFM01 (100 μM) treatment allows normal DSB repair in HR-defective ATMi-treated or HSC62 (BRCA2-defective) cells[1].RAD51 foci did not form following exo- or endo-inhibitor treatment (mirin or PFM01) in 1BR3 (WT) and HSC62 (BRCA2-defective) cells[1].PFM01 (100 μM) enhances non-homologous end-joining (NHEJ) in H1299 dA3 cells and reduces homologous recombination (HR) in U2OS DR-GFP cells[1].PFM01 substantially relieves the double-strand break (DSB) repair defect confers by mirin or PFM39 in irradiated G2 cells[1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 4 mg/mL (13.63 mM)
关键字: Inhibitor | derivative | MRE11 | PFM01 | NHEJ | Mirin | DSB | endonuclease | PFM 01 | N-alkylated | PFM-01 | inhibit
相关库: Bioactive Compounds Library Max | Inhibitor Library | DNA Damage & Repair Compound Library | Bioactive Compound Library
化合物PFM01 T8880信息由TargetMol中国为您提供,如您想了解更多关于化合物PFM01 T8880报价、型号、参数等信息,欢迎来电或留言咨询。
注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途