普林贝瑞 TQ0149
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
2 mg | 524684-52-4 | ¥449.00 | 询底价 |
1 mL | 524684-52-4 | ¥1,230.00 | 询底价 |
100 mg | 524684-52-4 | ¥6,870.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Prinaberel
描述: Prinaberel (ERB-041) is an effective and selective ERβ agonist and >200-fold selective for ERβ.
体外活性: Treatment with ERβ selective estrogen agonists liquiritigenin and ERB-041 reduced the ability to invade a reconstituted basement membrane and to migrate in response to the cellular stimulus [1]. Pretreatment the PMs with ERB-041 resulted in significant inhibition of LPS-induced iNOS expression and NF-kappaB activation by preventing its nuclear translocation [3].
体内活性: Tumor numbers and volume were reduced by 60% and 84%, respectively, in the Erb-041-treated group as compared with UVB (alone) control. This inhibition in tumorigenesis was accompanied by a decrease in proliferating cell nuclear antigen (PCNA), cyclin D1, VEGF, and CD31, and an increase in apoptosis [2].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 38 mg/mL (140.1 mM)
关键字: Prinaberel | ERB041 | ERB-041
相关产品: Chlorotrianisene | PROTAC ERRα ligand 2 | Ospemifene D4 | Endoxifen Z-isomer hydrochloride | Promestriene | Estradiol dipropionate | Altrenogest | Estradiol | NXT629 | (+)-Medicarpin
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途