化合物5HT6-ligand-1 T10053
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
1 mg | 1038988-11-2 | ¥1,380.00 | 询底价 |
50 mg | 1038988-11-2 | ¥9,360.00 | 询底价 |
100 mg | 1038988-11-2 | ¥12,400.00 | 询底价 |
10 mg | 1038988-11-2 | ¥4,670.00 | 询底价 |
5 mg | 1038988-11-2 | ¥3,340.00 | 询底价 |
25 mg | 1038988-11-2 | ¥6,900.00 | 询底价 |
Product Introduction
Bioactivity
英文名: 5HT6-ligand-1
描述: 5HT6-ligand-1 是一种具有口服活性的 5-HT6 受体配体 (Ki = 1.43 nM)。
体内活性: 5HT6-ligand-1(10 mg/kg) reverses the time delay-induced memory deficit and improves cognitive ability. 5HT6-ligand-1 shows an oral t1/2 of 3.17 h, a Cmax of 60 ng/mL, an exposure of 217 ng h/mL, and a bioavailability of 29%. Intravenous administration of 5HT6-ligand-1 exhibits a clearance of 220 mL/min/kg and a volume of distribution of 32.6 L/kg[1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 10 mg/mL (22.3 mM)
关键字: 5HT6-ligand-1 | 5HT6 ligand 1 | 5HT-6-ligand-1 | 5HT6ligand1
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相关库: Neurotransmitter Receptor Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | GPCR Compound Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途