化合物 T10360 T10360
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 220051-79-6 | ¥11,700.00 | 询底价 |
50 mg | 220051-79-6 | ¥15,300.00 | 询底价 |
100 mg | 220051-79-6 | ¥19,500.00 | 询底价 |
Product Introduction
Bioactivity
英文名: AR-A 2
描述: AR-A 2 is a selective 5-HT1B receptor antagonist, with a high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM).
体外活性: AR-A 2 (AR-A000002) is a selective 5-HT1B receptor antagonist and shows an EC50 of 4.5 nM for the guinea pig 5-HT1B receptor. AR-A 2 also binds to the rat cortical 5HT1B/1D receptor (Ki: 20 nM), rat cortex 5-HT2A receptor (Ki: 339 nM), rat hippocampus 5-HT1A receptor (Ki: 3070 nM). In addition, AR-A 2 also exhibits an affinity for dopamine D2 (Ki: 330 nM) and α1-adrenoceptors (Ki: 490 nM).
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: ARA 2 | AR-A-000002 | AR-A000002 | AR-A 2 | AR A 2
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途