化合物 T12344L T12344L
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 2093401-85-3 | ¥10,600.00 | 询底价 |
100 mg | 2093401-85-3 | ¥17,500.00 | 询底价 |
50 mg | 2093401-85-3 | ¥13,800.00 | 询底价 |
Product Introduction
Bioactivity
英文名: OTS186935 trihydrochloride
描述: OTS186935 trihydrochloride is a protein methyltransferase inhibitor of SUV39H2(IC50 of 6.49 nM).
体外活性: OTS186935 trihydrochloride, revealed significant inhibition of tumor growth in mouse xenograft models using MDA-MB-231 breast cancer cells and A549 lung cancer cells without any detectable toxicity.??SUV39H2 inhibitors sensitize cancer cells to DOX by reduction of γ-H2AX levels in cancer cells
体内活性: OTS186935 trihydrochloride?exhibits growth suppressive effects in human cancer cell line derived xenograft models[1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: OTS 186935 | OTS-186935 Trihydrochloride | OTS 186935 Trihydrochloride | OTS186935 trihydrochloride | OTS186935 Trihydrochloride | OTS186935 | OTS-186935 trihydrochloride | OTS-186935
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途