(S)-特拉唑嗪 T12815
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
50 mg | 109351-33-9 | ¥7,920.00 | 询底价 |
100 mg | 109351-33-9 | ¥12,500.00 | 询底价 |
25 mg | 109351-33-9 | ¥5,970.00 | 询底价 |
1 mL | 109351-33-9 | ¥2,280.00 | 询底价 |
2 mg | 109351-33-9 | ¥1,170.00 | 询底价 |
5 mg | 109351-33-9 | ¥1,980.00 | 询底价 |
Product Introduction
Bioactivity
英文名: (S)-Terazosin
描述: (S)-Terazosin is an active S-enantiomer of Terazosin. (S)-Terazosin is a potent and high-affinity antagonist of α-adrenoceptor(α1a, α1b and α1d-adrenoceptor with Ki values of 3.91 nM, 0.79 nM and 1.16 nM, respectively).
体外活性: (S)-Terazosin and its enantiomers show high and apparently equal affinity for subtypes of α1-adrenoceptors, and showed potent α1-adrenoceptors antagonist in isolated tissues, with the enantiomers approximately equipotent to the racemate at each α1-adrenoceptor subtype. At α2b sites, (R)-Terazosin binds less potently than either the (S)-Terazosin or racemate.
体内活性: (S)-Terazosin shows α2B receptor antagonist at rat atrial(pEC30 of 6.93). (s)-Terazosin shows antagonism of at rat vas deferens α1A and α2A receptor with pA2 values of 8.3 and 6.12, respectively.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 150 mg/mL (387.17 mM)
关键字: (S) Terazosin | (S)Terazosin | Terazosin
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途