化合物Adenosine A1 receptor activator T62 T14127
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
1 mg | 40312-34-3 | ¥1,190.00 | 询底价 |
500 mg | 40312-34-3 | ¥25,800.00 | 询底价 |
1 mL | 40312-34-3 | ¥2,730.00 | 询底价 |
25 mg | 40312-34-3 | ¥7,150.00 | 询底价 |
10 mg | 40312-34-3 | ¥4,630.00 | 询底价 |
100 mg | 40312-34-3 | ¥12,800.00 | 询底价 |
50 mg | 40312-34-3 | ¥9,630.00 | 询底价 |
5 mg | 40312-34-3 | ¥3,230.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Adenosine A1 receptor activator T62
描述: Adenosine A1 receptor activator T62 是腺苷 A1 受体的变构增强剂,有镇痛作用。
动物实验: Intrathecal T62 of Male SpragueDawley rats (250 g) after paw incision surgery with the dose of 0.3 μg, 0.5 μg, 1 μg, and 3 μg, produced a dose-dependent antihypersensitivity effect, with no effect on ambulation or activity level. The ED40 (95% confidence interval) for T62 was 0.77 (0.63-0.91) microg.
体内活性: Adenosine A1 receptor activator T62 (0.3-3 μg; intrathecal administration; male SpragueDawley rats) treatment produces a dose-dependent antihypersensitivity effect. However it has no effect on ambulation or activity level[1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 75 mg/ml (257.03 mM)
关键字: allosteric | Inhibitor | P1 receptor | adenosine | hypersensitivity | Adenosine Receptor | α2-adrenoceptors | antihypersensitivity | intrathecal | Enhancer | neuropathic | Adenosine A-1 receptor activator T62 | Adenosine A1 receptor activator T62 | inhibit
相关产品: Taminadenant | CPI-444 | Regadenoson | CHEMBL241987 | CCPA | SDZ WAG 994 | LAS101057 | 5-Iodotubercidin | BAY 60-6583 | MRS-1706
相关库: Drug Repurposing Compound Library | Neurotransmitter Receptor Compound Library | ReFRAME Related Library | Anti-Cancer Drug Library | Clinical Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | GPCR Compound Library | Anti-Cancer Clinical Compound Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途