化合物AR-C155858 T14316
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
100 mg | 496791-37-8 | ¥10,900.00 | 询底价 |
10 mg | 496791-37-8 | ¥3,690.00 | 询底价 |
25 mg | 496791-37-8 | ¥5,960.00 | 询底价 |
1 mL | 496791-37-8 | ¥2,570.00 | 询底价 |
50 mg | 496791-37-8 | ¥8,250.00 | 询底价 |
1 mg | 496791-37-8 | ¥861.00 | 询底价 |
5 mg | 496791-37-8 | ¥2,480.00 | 询底价 |
Product Introduction
Bioactivity
英文名: AR-C155858
描述: AR-C155858 是单羧酸转运蛋白 MCT1 和 MCT2 的抑制剂,Ki 分别为2.3和 10 nM。
体外活性: AR-C155858 (10 nM-100 nM) inhibits MCT1/MCT2 C-terminal chimaeras[1]. AR-C155858 inhibits MCT1 expressed in Xenopus oocytes in a time- and concentration-dependent manner[2]. AR-C155858 inhibits MCT2, and the 70% inhibition seen at 10 nM is followed by a gradually increasing inhibition which can only be explained by a Ki value of significantly less than 10 nM.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 40 mg/mL (86.67 mM)
关键字: inhibit | Inhibitor | AR-C-155858 | AR-C 155858 | Monocarboxylate Transporter | AR-C155858 | ARC155858 | AR C155858
相关产品: Niflumic acid | 7ACC1 | α-Cyano-4-hydroxycinnamic acid | AZD0095 | D-Phenylalanine | VB124 | Lactate transportor 1 | 7ACC2 | BAY-8002 | AZD3965
相关库: Ion Channel Inhibitor Library | Anti-Cancer Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Inhibitor Library | NO PAINS Compound Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途