化合物CCT129957 T14903

Product Introduction
Bioactivity


英文名: CCT129957

描述: CCT129957 是一种新型有效的磷脂酶 C-γ (PLC-γ) 抑制剂，IC50 约为 3 μM，GC50 为 15 μM。CCT129957 具有抗癌活性，在鳞状细胞中抑制 Ca2+ 的释放。

体外活性: The left phenyl group is situated within a hydrophobic pocket formed by various amino acids. The predicted binding mode of CCT129957 exhibits a robust hydrogen bonding pattern and hydrophobic contacts[1].CCT129957 inhibits the growth of renal UO-31 and breast T-47D cancer cells by approximately 60-70%[2].

存储条件: store at low temperaturePowder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 50 mg/mL (161.64 mM)


关键字: CCT 129957 | CCT129957 | CCT-129957

相关产品: Nexopamil | FS-2 | Ziconotide Acetate (107452-89-1 free base) | Ethyl cinnamate | Bryonolic acid | Fendiline hydrochloride | Nicardipine hydrochloride | Devapamil | ω-Tbo-IT1 | Maurocalcine

相关库: Membrane Protein-targeted Compound Library | Inhibitor Library

化合物CCT129957 T14903信息由TargetMol中国为您提供，如您想了解更多关于化合物CCT129957 T14903报价、型号、参数等信息，欢迎来电或留言咨询。

注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途