化合物 T15147 T15147
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
2 mg | 328104-79-6 | ¥819.00 | 询底价 |
100 mg | 328104-79-6 | ¥10,800.00 | 询底价 |
50 mg | 328104-79-6 | ¥6,990.00 | 询底价 |
25 mg | 328104-79-6 | ¥5,380.00 | 询底价 |
Product Introduction
Bioactivity
英文名: DNMDP
描述: DNMDP is a phosphodiesterase 3A inhibitor with clear cell-selective cytotoxicity. DNMDP binding to PDE3A promotes interaction between PDE3A and Schlafen 12.
体外活性: DNMDP (0-1000 μM; 48 hours) displays clear cell-selective cytotoxicity. HeLa cells undergo apoptosis upon DNMDP treatment, indicates by caspase activity detected by a caspase-sensitive luciferase assay and by PARP cleavage. DNMDP (100 nM) specifically inhibits both PDE3A and PDE3B, but it weakly inhibits PDE10. It also had little or no detectable effect on other phosphodiesterases.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: DNMDP
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途