化合物Eleclazine hydrochloride T15207
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 1448754-43-5 | ¥5,870.00 | 询底价 |
10 mg | 1448754-43-5 | ¥3,630.00 | 询底价 |
1 mg | 1448754-43-5 | ¥913.00 | 询底价 |
1 mL | 1448754-43-5 | ¥2,690.00 | 询底价 |
50 mg | 1448754-43-5 | ¥8,150.00 | 询底价 |
100 mg | 1448754-43-5 | ¥10,900.00 | 询底价 |
5 mg | 1448754-43-5 | ¥2,450.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Eleclazine hydrochloride
描述: Eleclazine hydrochloride (GS 6615 hydrochloride) 是新型 Na+电流抑制剂,IC50是0.7 uM。
体外活性: Inhibition by GS-6615 of ATX-II enhanced late INa is potently correlated with shortening of myocyte APD and isolated heart MAPD[1]. Eleclazine hydrochloride inhibits ATX-II enhanced late INa in ventricular myocytes, shorten the ATX-II induced prolongation of APD, MAPD, QT interval. It also decreased spatiotemporal dispersion of repolarization and ventricular arrhythmias. Selective inhibition of cardiac late INa with eleclazine hydrochloride confers dual protection against vulnerability to ischemia-induced AF. That decreases atrial and ventricular repolarization abnormalities before and during adrenergic stimulation without negative inotropic effects. [2]
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 100 mg/mL (221.32 mM)
关键字: Inhibitor | Eleclazine | GS-6615 | GS6615 | porcine | Eleclazine Hydrochloride | Sodium Channel | KcsA | Eleclazine hydrochloride | Na+ channels | inhibit | Na channels | epinephrine | Potassium Channel | GS6615 Hydrochloride | GS 6615 Hydrochloride | hiPSC | atrial premature beats | GS 6615 | GS-6615 Hydrochloride | cardiac arrhythmias
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相关库: Drug Repurposing Compound Library | Anti-Cancer Drug Library | Clinical Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Anti-Cancer Clinical Compound Library | Anti-Cardiovascular Disease Compound Library | NO PAINS Compound Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途