化合物AMN 082 dihydrochloride T21935
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
10 mg | 97075-46-2 | ¥1,438.00 | 询底价 |
Product Introduction
Bioactivity
英文名: AMN082
描述: AMN082 (AMN 082 dihydrochloride) 是可口服,可透过血脑屏障的选择性mGluR7激动剂,通过跨膜区的变构位点直接激活受体信号,具有抗抑郁作用。
体外活性: AMN082 inhibited 4-aminopyridine-evoked glutamate release and this phenomenon was blocked by the metabotropic glutamate mGlu7 receptor antagonist MMPIP.?Moreover, western blot analysis and immunocytochemistry confirmed the presence of presynaptic metabotropic glutamate mGlu7 receptor proteins.?The effect of AMN082 on the 4-aminopyridine-evoked release of glutamate was prevented by chelating the extracellular Ca2+ ions and the vesicular transporter inhibitor.[1]
体内活性: 动物预先处理较低剂量的AMN082(1.25-5.0 mg/kg,腹腔注射),在每次可卡因或吗啡注射前30分钟,或在重复给药期间及可卡因或吗啡挑战前,能剂量依赖性地减弱可卡因或吗啡引起的运动敏感化的发展和表达。[2]
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: inhibit | Inhibitor | AMN082 | allosteric | mGluR | AMN 082 Dihydrochloride | hormone | oral | Metabotropic glutamate receptors | stress | sensitization | AMN-082 | AMN082 Dihydrochloride | AMN 082 | locomotor | blood-brain | AMN-082 Dihydrochloride | barrier
相关产品: SIB-1757 | VU 0285683 | NPS2390 | MMPIP hydrochloride | CBiPES hydrochloride | LY404039 | pep2-EVKI acetate(1315378-67-6 free base) | ADX-47273 | DMeOB | Xanthurenic Acid
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途