化合物Guanabenz hydrochloride T21957

Product Introduction
Bioactivity


英文名: Guanabenz hydrochloride

描述: Guanabenz hydrochloride (NE56490) 是一种具有降血压作用的口服活性 α2-肾上腺素受体激动剂。

体内活性: Maximum concentrations of guanabenz hydrochloride in plasma (1.2 to 5.2 ng/ml) reached 2 to 5 hours after administration of capsules containing 16 or 32 mg of 14C-labelled guanabenz hydrochloride. Guanabenz hydrochloride was 90% bound to human plasma proteins. Guanabenz hydrochloride competed for imidazoline I2-binding sites in brown adipose tissue with Ki of 97 nM.

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 55 mg/ml (205.58 mM)


关键字: inhibit | Guanabenz hydrochloride | antiparasitic | Guanabenz Hydrochloride | NE-56490 | Inhibitor | Beta Receptor | NE 56490 | Guanabenz | Parasite | Adrenergic Receptor | antihypertensive | high blood pressure

相关产品: Pardoprunox hydrochloride | Spiroxatrine | Indacaterol maleate | Quinine HCl | ST 91 | Bedoradrine | Metaproterenol hemisulfate | Ketanserin tartrate | Tamsulosin hydrochloride | KUL-7211 racemate

相关库: Adrenergic Receptor-Targeted Compound Library | Drug Repurposing Compound Library | Anti-Neurodegenerative Disease Compound Library | Anti-Cancer Drug Library | Clinical Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | GPCR Compound Library | Anti-Cancer Clinical Compound Library | Anti-Cancer Approved Drug Library

化合物Guanabenz hydrochloride T21957信息由TargetMol中国为您提供，如您想了解更多关于化合物Guanabenz hydrochloride T21957报价、型号、参数等信息，欢迎来电或留言咨询。

注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途