半胆碱基-3 T2227

Product Introduction
Bioactivity


英文名: Hemicholinium 3

描述: Hemicholinium 3 是一种竞争性的、高亲和力的胆碱转运蛋白 (HACU) 抑制剂，Ki=25 nM。它是一种神经肌肉阻滞剂，能够抑制乙酰胆碱 (ACh)的合成和释放。它抑制Epibatidine 诱发的收缩和 [3H] 乙酰胆碱释放，IC50分别为 897 nM 和 693 nM。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 50 mg/mL (87.05 mM)


关键字: HACU | Choline | receptor | system | Hemicholinium dibromide | Inhibitor | transporter | Hemicholinium 3 | ACh | Nicotinic | Hemicholinium3 | inhibit | nervous | Enteric | neuromuscular | acetylcholine | Cholinesterase (ChE)

相关产品: 1-[10-(pyridin-1-ium-1-yl)decyl]pyridin-1-ium dibromide | SEW06622 | Minaprine | Histone acetyltransferase p300 Inhibitor 4c | Ethyl (triphenylphosphoranylidene) acetate | kuwanon G | Neoeriocitrin | Isomerazin | 1-Naphthyl acetate | Questin

相关库: Anti-Neurodegenerative Disease Compound Library | Neurotransmitter Receptor Compound Library | ReFRAME Related Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | Inhibitor Library | NO PAINS Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途