Z-因多昔芬 T2280
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
50 mg | 112093-28-4 | ¥2,320.00 | 询底价 |
5 mg | 112093-28-4 | ¥528.00 | 询底价 |
1 mg | 112093-28-4 | ¥228.00 | 询底价 |
10 mg | 112093-28-4 | ¥690.00 | 询底价 |
2 mg | 112093-28-4 | ¥326.00 | 询底价 |
1 mL | 112093-28-4 | ¥588.00 | 询底价 |
25 mg | 112093-28-4 | ¥1,450.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Endoxifen (Z-isomer)
描述: Endoxifen Z-isomer (EDX)是 Tamoxifen 重要的代谢产物,在表达 ERα的乳腺癌细胞中发挥抗雌激素作用。它以浓度依赖的方式抑制 hERG, IC50值为1.6μM。
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 45 mg/mL (120.48 mM)
关键字: Potassium Channel | Endoxifen | Endoxifen (Z-isomer) | Endoxifen (Zisomer) | Endoxifen (Z isomer) | Inhibitor | KcsA | inhibit | Z-isomer | Estrogen Receptor/ERR
相关产品: 14-3-3σ/ERα stabilizer-1 | Mestranol | Estetrol | Camizestrant | Endoxifen Z-isomer hydrochloride | Erteberel | G36 | Elacestrant | N-Desmethyltamoxifen hydrochloride | Estriol
相关库: JAK-STAT Compound Library | Drug Repurposing Compound Library | Anti-Prostate Cancer Compound Library | Anti-Cancer Drug Library | Membrane Protein-targeted Compound Library | Anti-Lung Cancer Compound Library | Kinase Inhibitor Library | Inhibitor Library | Anti-Cancer Clinical Compound Library | Tyrosine Kinase Inhibitor Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途