化合物GSK-LSD1 dihydrochloride T2315

Product Introduction
Bioactivity


英文名: GSK-LSD1 dihydrochloride

描述: GSK-LSD1 dihydrochloride (GSK-LSD1 2HCl) 是一种特异性不可逆的 LSD1 抑制剂(IC50: 16 nM)。GSK-LSD1 dihydrochloride 对 LSD1 的选择性是其他密切相关的 FAD 利用酶（即 MAO-A、LSD2、MAO-B）的 1000 倍以上。

体外活性: GSK-LSD1 induces gene expression changes in cancer cell lines with average EC50 of < 5 nM and inhibits cancer cell line growth with average EC50 of < 5 nM. [1]

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 4.23 mg/mL (14.63 mM)
H2O : 10 mg/mL (34.57 mM)


关键字: GSK LSD1 dihydrochloride | GSK-LSD1 Dihydrochloride | Monoamine Oxidase | GSK-LSD-1 dihydrochloride | Inhibitor | inhibit | MAO | GSKLSD1 dihydrochloride | Histone Demethylase | GSK-LSD1

相关产品: Eicosapentaenoic Acid | PFI-90 | TAK-418 | NCD38 TFA | GSK467 | GSK 690 Hydrochloride | IOX1 | JMJD7-IN-1 | GSK2879552 2HCl (1401966-69-5(free base)) | ML324

相关库: Anti-Aging Compound Library | Bioactive Compounds Library Max | Antidepressant Compound Library | Inhibitor Library | Epigenetics Compound Library | Stem Cell Differentiation Compound Library | Methylation Compound Library | Reprogramming Compound Library | Histone Modification Compound Library | Chromatin Modification Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途