化合物VU 10010 T23513

Product Introduction
Bioactivity


英文名: VU10010

描述: VU10010 (VU 10010) 是一种高度选择性的M4mAChR 变构增强剂，EC50为 400 nM。它与 M4mAChR 的变构位点结合，增强与 G 蛋白偶联，增加对乙酰胆碱的亲和力，还会增加卡巴胆碱引起的兴奋性传导抑制。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: Ethanol : < 1 mg/mL (insoluble or slightly soluble)
DMSO : < 34.59 mg/mL


关键字: hippocampus | synapses | acetylcholine | allosteric | excitatory | transmission | mAChR | Muscarinic acetylcholine receptor | carbachol | Inhibitor | inhibit | proteins | depression | VU-10010 | VU10010

相关产品: Donepezil Hydrochloride | Buxbodine B | GNF-7 | Lucidadiol | OXOMEMAZINE | Glycopyrrolate | YM-58790 | Gallamine triethiodide | YM17E | VU0357017 hydrochloride

相关库: Anti-Neurodegenerative Disease Compound Library | Neurotransmitter Receptor Compound Library | Anti-Parkinson's Disease Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | Anti-Alzheimer's Disease Compound Library | NO PAINS Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途