化合物PNU 282987 T2422
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
1 mg | 123464-89-1 | ¥189.00 | 询底价 |
1 mL | 123464-89-1 | ¥679.00 | 询底价 |
100 mg | 123464-89-1 | ¥3,720.00 | 询底价 |
25 mg | 123464-89-1 | ¥1,170.00 | 询底价 |
50 mg | 123464-89-1 | ¥1,950.00 | 询底价 |
10 mg | 123464-89-1 | ¥617.00 | 询底价 |
5 mg | 123464-89-1 | ¥383.00 | 询底价 |
Product Introduction
Bioactivity
英文名: PNU-282987
描述: PNU 282987 是一种选择性 α7 烟碱型乙酰胆碱受体 (α7 nAChR) 激动剂,Ki 为 26 nM。
激酶实验: Kinase inhibition assays : Kinase inhibition is measured by the use of radiometric assays conducted by Kinase Profiler service. Briefly, in the presence or absence of SKLB1002, VGFR2 (5–10 mU) is incubated in 25-μL reaction solution containing 8 mmol/L 3-(N-morpholino)propanesulfonic acid (MOPS), pH 7.0, 0.2 mmol/L EDTA, 0.33 mg/mL myelin basic protein, 10 mmol/L Mg acetate, and γ-[33P]ATP. After incubation for 40 minutes at room temperature, the reaction is stopped and 10 μL of the reaction solution is then spotted onto a P30 filtermat and washed 3 times for 5 minutes in 75 mmol/L phosphoric acid and once in methanol prior to scintillation counting.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 50 mg/mL (166 mM)
关键字: nAChR | PNU-282987 | Inhibitor | PNU282987 | Nicotinic acetylcholine receptors | inhibit | PNU 282987
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途