化合物AZD1940 T30252

Product Introduction
Bioactivity


英文名: AZD1940

描述: AZD1940 (UNII-0J0035E9FT)是一种高亲和力的大麻素CB(1)/CB(2)受体激动剂，具有口服活性，应用于口面疼痛的研究。

体外活性: AZD1940 binds with high affinity to human, rat and mouse CB1 and CB2 receptors and displays full agonism at both receptors in all three species[1].

体内活性: 口服给予人体后，AZD1940 800 mg的平均最大血浆浓度（Cmax）为9.3 nmol/L。在剂后八小时内，AZD1940的平均浓度为236 nmol·h/L[1]。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 90.0 mg/mL (217.6 mM)


关键字: AZD1940

相关产品: PSB-SB-487 | Drinabant | PrNMI | Hemopressin (human, mouse) acetate | 2-Arachidonoylglycerol | CB2R agonist 2 | N-Oleoyl glycine | OMDM-5 | Otenabant hydrochloride | β-Caryophyllene

相关库: Drug Repurposing Compound Library | Anti-Cancer Drug Library | Clinical Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | Anti-Cancer Clinical Compound Library | GPCR Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途