rac-trans-4-hydroxy Glyburide T35635
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
1 mg | 23155-00-2 | ¥1,970.00 | 询底价 |
Product Introduction
Bioactivity
英文名: rac-trans-4-hydroxy Glyburide
描述: rac-trans-4-hydroxy Glyburide is an active metabolite of the SUR1/Kir6.2 sulfonylurea inhibitor glyburide .1,2It is formed from glyburide by the cytochrome P450 (CYP) isoforms CYP2C8 and CYP2C9.1rac-trans-4-hydroxy Glyburide inhibits glyburide binding to rat brain synaptosomes at the high and low affinity sites of SUR1/Kir6.2 with IC50values of 0.95 and 100 nM, respectively.2
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: Methanol : Slightly soluble
DMSO : Slightly soluble
关键字: ractrans4hydroxy Glyburide | rac trans 4 hydroxy Glyburide | rac-trans-4-hydroxy Glyburide
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途