CCG258208 hydrochloride T35875

Product Introduction
Bioactivity


英文名: CCG258208 hydrochloride

描述: GRKs-IN-1 hydrochloride, Compound 14as, has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50=130 nM) and GRK5 (IC50=7.1 μM).GRKs-IN-1 hydrochloride is a derivative 14as of paroxetine, shows a 100-fold improvement in cardiomyocyte contractility assays over paroxetine[1].

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: H2O : 50 mg/mL (102.26 mM)
DMSO : 250 mg/mL (511.31 mM)


关键字: CCG 258208 Hydrochloride | CCG258208 hydrochloride | CCG-258208 Hydrochloride | CCG-258208 hydrochloride | CCG258208 Hydrochloride

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途