N-去甲基西地那非 T36061
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
1 mg | 139755-82-1 | ¥413.00 | 询底价 |
500 mg | 139755-82-1 | ¥13,500.00 | 询底价 |
50 mg | 139755-82-1 | ¥4,680.00 | 询底价 |
1 mL | 139755-82-1 | ¥1,090.00 | 询底价 |
100 mg | 139755-82-1 | ¥6,680.00 | 询底价 |
25 mg | 139755-82-1 | ¥3,160.00 | 询底价 |
5 mg | 139755-82-1 | ¥946.00 | 询底价 |
10 mg | 139755-82-1 | ¥1,580.00 | 询底价 |
Product Introduction
Bioactivity
英文名: N-Desmethyl Sildenafil
描述: N-Desmethyl Sildenafil (UK-103,320) (Desmethylsildenafil) 是Sildenafil的主要代谢物,是一种强效的磷酸二酯酶类型5(PDE5)抑制剂。
体外活性: N-Desmethyl Sildenafil increases the amplitude of electroretinogram (ERG) recorded from the dark-adapted isolated rat retina, most probably through the enhancement of the photoreceptor cell response[1]. The formation of N-Desmethyl Sildenafil is examined using CYP3A supersomes co-expressing human P450 oxidoreductase and cytochrome b5. N-Desmethyl Sildenafil is catalyzed by CYP3A4, CYP3A5, and to a lesser extent by CYP3A7[2].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMF : 5 mg/mL
DMSO:PBS (pH 7.2)(1:5) : 0.15 mg/mL
DMSO : 225 mg/mL (488.5 mM)
关键字: N-Desmethyl Sildenafil
相关产品: p,p'-DDE | RPR132595A hydrochloride | CLOZAPINE N-OXIDE | GS-443902 | Hydroxy Dimetridazole | N-Desmethyl imatinib | Urolithin A | AST5902 mesylate(2412155-74-7 free base) | Desmethyl Erlotinib hydrochloride | Desmethyl Erlotinib
N-去甲基西地那非 T36061信息由TargetMol中国为您提供,如您想了解更多关于N-去甲基西地那非 T36061报价、型号、参数等信息,欢迎来电或留言咨询。
注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途