化合物[Orn8]-Urotensin II acetate T37527L

Product Introduction
Bioactivity


英文名: [Orn8]-Urotensin II acetate

描述: [Orn8]-Urotensin II acetate 是一种 Urotensin 受体配体和 Urotensin 受体的部分激动剂。

体内活性: [Orn8]-Urotensin II acetate behaves as a full agonist (pEC50 approximately equal 8) at both human and rat UT receptors in the FlipR calcium assay eliciting similar maximal effects as the natural ligand U-II. On the contrary, in the rat aorta bioassay, [Orn8]-Urotensin II acetate behaves as a competitive and selective antagonist (pA2 = 6.56) showing however a small but consistent residual agonist activity[2].

存储条件: keep away from moisturePowder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 14.35 mg/mL (10 mM)


关键字: [Orn8]Urotensin II acetate | [Orn8]-Urotensin II Acetate | [Orn8] Urotensin II acetate | [Orn-8]-Urotensin II acetate(479065-85-5 Free base)

相关产品: TUG-499 | APD668 | 2-Oleoylglycerol | GPR120 Agonist 3 | Fasiglifam | 4-CMTB | CAY10471 Racemate | (2-{[2-(2-fluorophenoxy)ethyl]sulfanyl}-1H-benzimidazol-1-yl)acetic acid | PU-WS13 hydrobromide | TUG-469

相关库: Membrane Protein-targeted Compound Library | Peptide Compound Library

化合物[Orn8]-Urotensin II acetate T37527L信息由TargetMol中国为您提供，如您想了解更多关于化合物[Orn8]-Urotensin II acetate T37527L报价、型号、参数等信息，欢迎来电或留言咨询。

注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途