Squarunkin A hydrochloride T37597
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
50 mg | 2253744-55-5 | ¥13,800.00 | 询底价 |
100 mg | 2253744-55-5 | ¥17,500.00 | 询底价 |
25 mg | 2253744-55-5 | ¥10,600.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Squarunkin A hydrochloride
描述: Squarunkin A hydrochloride 是一种有效的选择性UNC119-货物相互作用抑制剂。Squarunkin A hydrochloride 选择性地抑制Src 激酶 N 末端的肉豆蔻酰化肽与 UNC119A 的结合,IC50 值为 10 nm。Squarunkin A hydrochloride 会干扰细胞中Src 激酶的活化。
体外活性: Squarunkin A (2.5 μM, 0.625 μM, 0.078 μM, and 0.01 μM) treatment results in a concentration-dependent reduction of Src phosphorylation [1]. Squarunkin A does not target the lipoprotein-binding sites of other lipoprotein chaperones, such as PDE6d, AIPL1, and RhoGDI, which bind S-prenylated proteins. Squarunkin A binds to UNC119 in cell lysate and interferes with Src activation [1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : Soluble
关键字: Squarunkin A hydrochloride | Squarunkin A Hydrochloride
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途