Salvinorin A Propionate T38055

Product Introduction
Bioactivity


英文名: Salvinorin A Propionate

描述: Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM. It inhibits adenylate cyclase (EC50 = 4.7 nM) in HEK293 cells transfected with human KOR. It is selective for KORs over μ, δ, and ORL-1 opioid receptors and has no effect at serotonin, dopamine, muscarinic, or adrenergic receptors. In mice, salvinorin A propionate (13 μg, i.c.v.) reduces nociceptive responses in a radiant heat tail-flick assay, though not as potently as salvinorin A .

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMF:PBS(pH 7.2)(1:1) : 0.5 mg/mL
DMF : 2 mg/mL
Acetonitrile : 1 mg/mL
DMSO : 1 mg/mL


关键字: Salvinorin A Propionate

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途