SPOP-IN-6b hydrochloride T39593
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 2136270-68-1 | ¥10,600.00 | 询底价 |
Product Introduction
Bioactivity
英文名: SPOP-IN-6b hydrochloride
描述: SPOP-IN-6b hydrochloride is a highly effective inhibitor of speckle-type POZ protein (SPOP), exhibiting an IC50 value of 3.58 μM.
体外活性: SPOP-IN-6b shows IC 50 s of 2-10.2 μM for A498, Caki-2, Ketr-3, 769-P, 0S-RC-2 and 786-0 cells[1]. SPOP-IN-6b (0.1-3.0 μM; 10 hours) can suppress SPOP activity, and then increase suppression cancer substrate protein PTEN and DUSP7 content[1].
体内活性: SPOP-IN-6b (40-80 mg/kg; intraperitoneal injection; daily; for 25 days; nude mice) can slow down the growth of tumour by suppressing SPOP[1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: SPOP-IN-6b Hydrochloride | SPOPIN6b hydrochloride | SPOP IN 6b hydrochloride
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途