BCR-ABL-IN-3 T39732
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 2240191-12-0 | ¥10,600.00 | 询底价 |
Product Introduction
Bioactivity
英文名: BCR-ABL-IN-3
描述: BCR-ABL-IN-3 is a highly effective and irreversibly binding inhibitor of Bcr-Abl, displaying a remarkable potency with an IC50 value of ≤100 nM for Ba/F3 Bcr-Abl T3151. This compound exhibits significant anti-cancer activity.
体内活性: BCR-ABL-IN-3 (compound 7; 15 mg/kg; twice a day; for 19 days) has good antitumor effect in female NOD/SCID mice of 7-8 weeks weighing 21.8 g with Ba/F 3 Bcr-Abl T3151 cells[1]. BCR-ABL-IN-3 (2 mg/kg for IV or 20mg/kg for PO) has a C max of 5485 ng/mL and an AUC of 5450 h?ng/mL for IV in male Sprague Dawley rats of 7-8 weeks old weighing 210 g[1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: BCR-ABL-IN-3 | BCRABLIN3 | BCR ABL IN 3
BCR-ABL-IN-3 T39732信息由TargetMol中国为您提供,如您想了解更多关于BCR-ABL-IN-3 T39732报价、型号、参数等信息,欢迎来电或留言咨询。
注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途