塞拉菌素 T4059

Product Introduction
Bioactivity


英文名: Selamectin

描述: Selamectin (UK-124114) 是半合成的大环内酯，是一种驱虫剂，可增强线虫中谷氨酸和 GABA 门控氯离子通道的开放。它还是抗寄生虫剂，可激活神经元和咽肌中的谷氨酸门控氯离子通道，以预防恶丝虫，淋巴丝虫和线虫感染。它还是 P-糖蛋白底物和抑制剂，IC50为 120 nM。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 90 mg/mL(116.9 mM)


关键字: Chloride Channel | MDR1 | P-glycoprotein | Multidrug resistance protein 1 | Parasite | UK 124114 | P-gp | ABCB1 | UK124114 | Cluster of differentiation 243 | Inhibitor | Pgp | Cl? Channels | Selamectin | inhibit | CD243

相关产品: R(+)-IAA-94 | Niflumic acid | ANO1-IN-1 | Shikonin | Flufenamic acid | Meticrane | T16Ainh-A01 | Ani9 | Adjudin | D-Alanine

相关库: Ion Channel Inhibitor Library | Drug Repurposing Compound Library | Anti-Cancer Compound Library | Anti-Cancer Drug Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Anti-Cancer Approved Drug Library | Anti-Parasitic Compound Library | NO PAINS Compound Library

塞拉菌素 T4059信息由TargetMol中国为您提供，如您想了解更多关于塞拉菌素 T4059报价、型号、参数等信息，欢迎来电或留言咨询。

注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途