柯因二甲醚 T5778

Product Introduction
Bioactivity


英文名: 5,7-DIMETHOXYFLAVONE

描述: 5,7-Dimethoxyflavone 是一种 Kaempferia parviflora 的主要成分，具有抗肿瘤、抗肥胖及抗炎活性。它对细胞色素 P450 (CYP) 3As 具有抑制作用，也是抗乳腺癌蛋白 (BCRP) 抑制剂。

体外活性: The best in vitro trypanocidal activity for T. brucei rhodesiense was exerted by 7,8-dihydroxyflavone (50% inhibitory concentration [IC50], 68 ng/ml), followed by 3-hydroxyflavone, rhamnetin, and 7,8,3',4'-tetrahydroxyflavone (IC50s, 0.5 microg/ml) and catechol (IC50, 0.8 microg/ml).?The activity against T. cruzi was moderate, and only Chrysin dimethylether and 3-hydroxydaidzein had IC50s less than 5.0 microg/ml.

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 50 mg/mL (177.12 mM)


关键字: anti-inflammatory | Cytochrome P450 | Anti-obesity | CYPs | 5,7 DIMETHOXYFLAVONE | inhibit | CYP3As | antineoplastic | BCRP | 5,7-DIMETHOXYFLAVONE | 5,7-Dimethoxyflavone | Inhibitor | 5,7DIMETHOXYFLAVONE

相关产品: 7-Hydroxyflavanone | Pyrolin | Isoschaftoside | 8-Epidiosbulbin E acetate | 4-Acetamidobenzenesulfonamide | 2'-Hydroxy-4'-methylacetophenone | Octahydrocurcumin | Quercimeritrin | Nevadensin | Sulfabrom

相关库: Selected Plant-Sourced Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Traditional Chinese Medicine Monomer Library | Anti-Cancer Active Compound Library | Natural Product Library for HTS | Metabolism Compound Library | Flavonoid Natural Product Library | NO PAINS Compound Library | Natural Product Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途