化合物 Chitin synthase inhibitor 1 T62068
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | 价格 | 操作 |
---|---|---|
100 mg | ¥17,500.00 | 询底价 |
25 mg | ¥10,600.00 | 询底价 |
50 mg | ¥13,800.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Chitin synthase inhibitor 1
描述: Chitin synthase inhibitor 1 是有效的、选择性的几丁质合酶 (CHS) 抑制剂,IC50值为0.12 mM。Chitin synthase inhibitor 1 强效抑制耐药真菌变体。
体外活性: Chitin synthase inhibitor 1 (compound 5a) shows broad-spectrum antifungal activity (MIC=4 μg/mL in Candidaalbicans (C. albicans) ATCC 76615 and Aspergillus fumigatus (A. fumigatus) GIMCC 3.19; MIC=8 μg/mL in Aspergillus flavus (A. flavus) ATCC 16870 and Crytococcusneoformans (C. neoformans) ATCC 32719) [1]. Chitin synthase inhibitor 1 shows antifungal activity against drug-resistant fungi variants (MIC=32 μg/mL in Fluconazoleresistant C.albicans ATCC 76615R, Fluconazole-resistant A.fumigatus GIMCC 3.19R, and Fluconazole-resistant C. neoformans ATCC 32719R, Micafunginresistant C.albicans ATCC 76615R’; MIC=16 μg/mL in Fluconazole-resistant A.flavus ATCC 16870R) [1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途