化合物 SAX-187 hydrochloride T69104

Product Introduction
Bioactivity


英文名: SAX-187 hydrochloride

描述: SAX-187 hydrochloride is a potent and selective 5-HT6 receptor agonist. SAX-187 hydrochloride possesses high affinity binding (2.2 and 4.8 nM, respectively) at the human 5-HT6 receptor and profile as full receptor agonists (SAX-187 hydrochloride: EC50=6.6 nM, Emax=93%). In the rat frontal cortex, acute administration of SAX-187 hydrochloride (3-30 mg/kg, subcutaneous (s.c.)) significantly increased extracellular GABA concentrations without altering the levels of glutamate or norepinephrine.

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

关键字: SAX-187 Hydrochloride | WAY181187 | WAY 181187 | WAY-181187 hydrochloride | WAY-181187 HCl | SAX 187 Hydrochloride | SAX187 Hydrochloride

化合物 SAX-187 hydrochloride T69104信息由TargetMol中国为您提供，如您想了解更多关于化合物 SAX-187 hydrochloride T69104报价、型号、参数等信息，欢迎来电或留言咨询。

注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途