(+/-)-双氮奋兴 T7341

Product Introduction
Bioactivity


英文名: Diclofensine

描述: Diclofensine (Ro 8-4650) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。

动物实验: In a controlled study, out-patients suffering from moderate to severe depression were treated with the objective of assessing the new drug's therapeutically effective dose range. Maprotiline was used as a reference drug: fourteen patients were assigned to receive diclofensine and thirteen to receive maprotiline in a double-blind design. Depending on tolerance and efficacy, they were treated for periods ranging from 5 to 150 days. Doses were titrated to the optimum[1].

体内活性: A controlled trial with diclofensine, a new psychoactive drug, in the treatment of depression[1].

存储条件: keep away from direct sunlight,store under nitrogen,store at low temperature,keep away from moisturePowder: -20°C for 3 years | In solvent: -80°C for 1 year

关键字: SLC6A3 | Inhibitor | DAT | Dopamine Transporter | Diclofensine | inhibit

相关产品: Atomoxetine hydrochloride | Perphenazine | 5,7-Dimethoxyluteolin | PF-00217830 | Fananserin | Piperacetazine | 9-FLUORENOL | Ansofaxine hydrochloride | GR 103691 | Diclofensine hydrochloride

(+/-)-双氮奋兴 T7341信息由TargetMol中国为您提供，如您想了解更多关于(+/-)-双氮奋兴 T7341报价、型号、参数等信息，欢迎来电或留言咨询。

注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途