呋拉茶碱 T7410

Product Introduction
Bioactivity


英文名: Furafylline

描述: Furafylline 是有选择性的人细胞色素P450IA2抑制剂(IC50:0.07 μM)。

体外活性: Furafylline是一种强效的、非竞争性抑制剂，专门针对人类肝脏微粒体部分中高亲和力的苯乙酮O-去乙基化酶活性进行抑制，该反应由P450IA2催化，其IC50值为0.07 microM[1]。

体内活性: Furafylline最初作为一种与theophylline[1]相比具有延长作用时间的支气管扩张剂被引入。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 12.5 mg/mL (48.03 mM)


关键字: Cytochrome P450 | inhibit | Inhibitor | CYPs | Furafylline

相关产品: CRTH2-IN-1 | Beta-Tetralone | Retrorsine | 2-Hydroxy-1-Methoxyaporphine | Alizarin | Avasimibe | K777 | EN3356 | Cedrol | Resveratroloside

相关库: Anti-Aging Compound Library | Anti-Cancer Compound Library | Anti-Metabolism Disease Compound Library | Bioactive Compounds Library Max | Human Metabolite Library | Inhibitor Library | Lipid Metabolism Compound Library | Metabolism Compound Library | NO PAINS Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途