[DPro10] Dynorphin A (1-11)acetate(猪） T76341L

Product Introduction
Bioactivity


英文名: [DPro10] Dynorphin A (1-11)acetate,porcine

描述: [DPro10] Dynorphin A (1-11)acetate,porcine 是一种高效的 κ-阿片受体激动剂，其 Ki 值为 0.13 nM。[DPro10] Dynorphin A (1-11), porcine 是一种 N-烷基化衍生物，具有镇痛活性。

体外活性: Porcine [DPro10] Dynorphin A (1-11) inhibits adenylyl cyclase activity in CHO cells expressing k-opioid receptors, with an IC50 value of 0.12 nM[1].

体内活性: Administered intracerebroventricularly (ICV), [DPro10] Dynorphin A (1-11), porcine, exhibits analgesic effects involving thermal cutaneous (tail-flick) and chemical visceral (acetic acid-induced writhing) stimuli, with known differential activation of mu and kappa receptors[2].

存储条件: store at low temperature,keep away from moisturePowder: -20°C for 3 years | In solvent: -80°C for 1 year

关键字: [DPro10] Dynorphin A acetate,porcine

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相关库: Anti-Neurodegenerative Disease Compound Library | Membrane Protein-targeted Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途