化合物Ipamorelin 2 Pivalic acid T7809L
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
2 mg | T7809L | ¥736.00 | 询底价 |
100 mg | T7809L | ¥5,680.00 | 询底价 |
10 mg | T7809L | ¥1,490.00 | 询底价 |
25 mg | T7809L | ¥2,680.00 | 询底价 |
50 mg | T7809L | ¥3,990.00 | 询底价 |
1 mg | T7809L | ¥496.00 | 询底价 |
5 mg | T7809L | ¥1,130.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Ipamorelin 2 Pivalic acid
描述: Ipamorelin 2 Pivalic acid (NNC-26-0161) 是一种生长激素释放肽,可诱导大鼠纵向骨生长。
体外活性: In vitro, ipamorelin released GH from primary rat pituitary cells with a potency and efficacy similar to GHRP-6 (ECs) = 1.3+/-0.4nmol/l and Emax = 85+/-5% vs 2.2+/-0.3nmol/l and 100%).?A pharmacological profiling using GHRP and growth hormone-releasing hormone (GHRH) antagonists clearly demonstrated that ipamorelin, like GHRP-6, stimulates GH release via a GHRP-like receptor[1]
体内活性: In pentobarbital anaesthetised rats, ipamorelin released GH with a potency and efficacy comparable to GHRP-6 (ED50 = 80+/-42nmol/kg and Emax = 1545+/-250ng GH/ml vs 115+/-36nmol/kg and 1167+/-120ng GH/ml).?In conscious swine, ipamorelin released GH with an ED50 = 2.3+/-0.03 nmol/kg and an Emax = 65+/-0.2 ng GH/ml plasma.?Again, this was very similar to GHRP-6 (ED50 = 3.9+/-1.4 nmol/kg and Emax = 74+/-7ng GH/ml plasma)[1].
存储条件: keep away from moisturePowder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 10 mM
关键字: Ipamorelin 2acetate(170851704(free base)) | Ipamorelin 2acetate(170851 70 4(free base)) | Ipamorelin 2 Pivalic acid
相关库: Drug Repurposing Compound Library | Clinical Compound Library | Bioactive Compounds Library Max | NO PAINS Compound Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途