化合物BYK204165 T7896

Product Introduction
Bioactivity


英文名: BYK204165

描述: BYK204165 (RT-017290) 是一种选择性PARP1抑制剂，对重组人 PARP1的pIC50值为 7.35，pKi 值为7.05。它对鼠 PARP-2的pIC50值为 5.38 ，其对 PARP1 的选择性比对 PARP2 高 100 倍。

体外活性: BYK204165 displayed 100-fold selectivity for PARP-1[1].

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 125 mg/mL (495.50 mM)


关键字: RT017290 | poly ADP ribose polymerase | BYK-204165 | Inhibitor | RT 017290 | BYK 204165 | PARP | antitumor | inhibit | BYK204165

相关产品: OUL35 | Rucaparib Phosphate | Buddlejasaponin IV | PARP-1-IN-4 | WAY-620473 | E7016 | Verbascoside | PARP1-IN-8  | AZ6102 | PARP10-IN-3

相关库: Anti-Aging Compound Library | Anti-Breast Cancer Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Epigenetics Compound Library | Anti-Pancreatic Cancer Compound Library | Anti-Cardiovascular Disease Compound Library | Covalent Inhibitor Library | NO PAINS Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途