盐酸屈他维林 T8787
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 985-12-6 | ¥1,450.00 | 询底价 |
1 mL | 985-12-6 | ¥547.00 | 询底价 |
500 mg | 985-12-6 | ¥8,790.00 | 询底价 |
10 mg | 985-12-6 | ¥747.00 | 询底价 |
1 mg | 985-12-6 | ¥218.00 | 询底价 |
5 mg | 985-12-6 | ¥495.00 | 询底价 |
50 mg | 985-12-6 | ¥2,660.00 | 询底价 |
100 mg | 985-12-6 | ¥3,930.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Drotaverine hydrochloride
描述: Drotaverine hydrochloride 是磷酸二酯酶 4 (PDE4)的抑制剂,也是 L 型电压依赖钙通道(L-VDCC)的阻滞剂,可阻断3',5'-环腺苷单磷酸的降解。它在体内有抗痉挛效果,但无抗胆碱能的效果。
体外活性: drotaverine not only relaxed the precontracted tracheal preparations but also decreased mediator-induced contraction.?These effects of drotaverine were concentration dependent, with a significantly higher potency on the KCl-induced response, than on either the histamine or methacholine induced one.?A similar result was noted for nifedipine.?The PDE inhibitor, theophylline, also relaxed the precontracted preparations but was ineffective on the mediator-induced contraction in a physiologically relevant concentration range.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 25 mg/mL (57.61 mM)
关键字: Ca2+ channels | Inhibitor | Drotaverine hydrochloride | Ca channels | inhibit | Drotaverine | Phosphodiesterase (PDE) | Drotaverine Hydrochloride | Calcium Channel
相关产品: Isopedicin | Thioquinapiperifil dihydrochloride | PF-00489791 | Nortadalafil | Ziritaxestat | WAY-313170 | Autotaxin-IN-1 | Acefylline | Kuraridine | Moracin M
相关库: Anti-Neurodegenerative Disease Compound Library | Drug Repurposing Compound Library | Human Metabolite Library | Inhibitor Library | Metabolism Compound Library | RO5 Drug-like Natural Product Library | Anti-Alzheimer's Disease Compound Library | Anti-Cardiovascular Disease Compound Library | NO PAINS Compound Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途