化合物Thioquinapiperifil二盐酸盐 T9773
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
100 mg | 204077-66-7 | ¥15,300.00 | 询底价 |
500 mg | 204077-66-7 | ¥29,700.00 | 询底价 |
10 mg | 204077-66-7 | ¥5,490.00 | 询底价 |
25 mg | 204077-66-7 | ¥8,480.00 | 询底价 |
50 mg | 204077-66-7 | ¥11,300.00 | 询底价 |
1 mL | 204077-66-7 | ¥4,410.00 | 询底价 |
1 mg | 204077-66-7 | ¥1,510.00 | 询底价 |
5 mg | 204077-66-7 | ¥3,830.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Thioquinapiperifil dihydrochloride
描述: Thioquinapiperifil dihydrochloride 是一种磷酸二酯酶(PDE-5)抑制剂(IC50: 0.074 nM),具有有效性、选择性和非竞争性,可用于研究性成熟。
体外活性: Thioquinapiperifil dihydrochloride (KF31327) (0.1-10 μM) inhibits platelet aggregation in a concentration-dependent manner. In the absence of nitroglycerin, higher concentrations of 1 and 10 μM of KF31327 are inhibits platelet aggregation in a concentration-dependent manner.[2] Thioquinapiperifil dihydrochloride (KF31327) shows a significant increase in cyclic GMP at 10 μM. After 5 min incubation, the mean cyclic GMP levels of KF31327-treated cells is 0.95±0.17 pmol/10 8 cells.[2]
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 112.5 mg/mL (215.7 mM)
关键字: KF 31327 | KF31327 | Thioquinapiperifil | Thioquinapiperifil Dihydrochloride
相关产品: Lirimilast | Saterinone | uk-50001 | Tofimilast | BC 11-38 | MY-5445 | Isoprenaline hydrochloride | Sulmazole | CM-675 | Triflusal
相关库: Bioactive Compounds Library Max | Inhibitor Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途