孕烯醇酮醋酸酯 TC0019

Product Introduction
Bioactivity


英文名: Pregnenolone acetate

描述: Pregnenolone acetate 是一种强大的神经类固醇，是各种类固醇激素（包括类固醇酮）的主要前体。它作为大麻素 CB1 受体的信号特异性抑制剂，抑制由 CB1 受体介导的四氢大麻酚 (THC) 的作用。它可以保护大脑免受大麻中毒。

体外活性: Pregnenolone likely acts as a signaling-specific negative allosteric modulator binding to a site distinct from that occupied by orthosteric ligands. Pregnenolone does not modify agonist binding but only agonist efficacy[1].

体内活性: Pregnenolone acetate is a powerful neurosteroid, the main precursor of various steroid hormones including steroid ketones.?It acts as a signaling-specific inhibitor of cannabinoid CB1 receptor, inhibits the effects of tetrahydrocannabinol (THC) that are mediated by the CB1 receptors. It?can protect the brain from cannabis intoxication[1].

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : Insoluble
H2O : Insoluble


关键字: 3beta-Hydroxy-5-pregnen-20-one Acetate | 3b-Hydroxy-5-pregnen-20-one Acetate | 3β-Hydroxy-5-pregnen-20-one Acetate | Pregnenolone acetate | Pregnenolone Acetate

相关产品: AM-1235 | JD-5037 | CB2 PET Radioligand 1 | (±)-Cannabichromene | Bay 59-3074 | Org 27569 | AM841 | ML192 | CB1 antagonist 2 | CB1 inverse agonist 1

相关库: RO5 Drug-like Natural Product Library

孕烯醇酮醋酸酯 TC0019信息由TargetMol中国为您提供，如您想了解更多关于孕烯醇酮醋酸酯 TC0019报价、型号、参数等信息，欢迎来电或留言咨询。

注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途